Development of the First Covalent Monopolar Spindle Kinase 1 (MPS1/TTK) Inhibitor

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Development of the First Covalent Monopolar Spindle Kinase 1 (MPS1/TTK) Inhibitor

Author: Serafim, Ricardo A. M.; Santiago, Andre da Silva; Schwalm, Martin P.; Hu, Zexi; dos Reis, Caio, V; Takarada, Jessica E.; Mezzomo, Priscila; Massirer, Katlin B.; Kudolo, Mark; Gerstenecker, Stefan; Chaikuad, Apirat; Zender, Lars; Knapp, Stefan; Laufer, Stefan; Counago, Rafael M.; Gehringer, Matthias
Tübinger Autor(en):
Serafim, Ricardo A. M.
Hu, Zexi
Kudolo, Mark
Gerstenecker, Stefan
Zender, Lars
Laufer, Stefan
Gehringer, Matthias
Published in: Journal of Medicinal Chemistry (2022), Bd. 65, H. 4, S. 3173-3192
Verlagsangabe: Amer Chemical Soc
Language: English
Full text: http://dx.doi.org/10.1021/acs.jmedchem.1c01165
ISSN: 0022-2623
DDC Classifikation: 540 - Chemistry and allied sciences
Dokumentart: Article
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